| Reaction Details |
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 | Report a problem with these data |
| Target | D(1A) dopamine receptor |
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| Ligand | BDBM50401950 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_886473 (CHEMBL2214284) |
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| Ki | 1400±n/a nM |
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| Citation |  Löber, S; Hübner, H; Buschauer, A; Sanna, F; Argiolas, A; Melis, MR; Gmeiner, P Novel azulene derivatives for the treatment of erectile dysfunction. Bioorg Med Chem Lett22:7151-4 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(1A) dopamine receptor |
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| Name: | D(1A) dopamine receptor |
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| Synonyms: | DRD1 | DRD1_PIG | Dopamine D1 receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 49269.92 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_1460140 |
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| Residue: | 446 |
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| Sequence: | MRTLNTSTMDGTGLVVERDFSFRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTN
FFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVD
RYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNVTSLG
KTTHNCDSSLSRTYAISSSLISFYIPVAIMIVTYTRIYRIAQKQIRRISALERAAVHAKN
CQTTAGNGNPAECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCMVPFCGS
GETKPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPTSTNAIET
VSINNNGAVVFSSHHEPRGSISKDCNLVYLIPHAVGSSEDLKKEEAGGIASPLEKLSPAL
SVILDYDTDVSLEKIQPITQNGQHPT
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| BDBM50401950 |
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| n/a |
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| Name | BDBM50401950 |
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| Synonyms: | CHEMBL2207634 |
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| Type | Small organic molecule |
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| Emp. Form. | C27H30N2O |
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| Mol. Mass. | 398.5399 |
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| SMILES | CCCC#Cc1cc(CN2CCN(CC2)c2ccccc2OC)c2cccccc12 |
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| Structure | 
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