| Reaction Details |
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 | Report a problem with these data |
| Target | Carnitine O-palmitoyltransferase 2, mitochondrial |
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| Ligand | BDBM50403031 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_887417 (CHEMBL2217026) |
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| IC50 | 4700±n/a nM |
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| Citation |  Ceccarelli, SM; Chomienne, O; Gubler, M; Arduini, A Carnitine palmitoyltransferase (CPT) modulators: a medicinal chemistry perspective on 35 years of research. J Med Chem54:3109-52 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Carnitine O-palmitoyltransferase 2, mitochondrial |
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| Name: | Carnitine O-palmitoyltransferase 2, mitochondrial |
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| Synonyms: | CPT II | CPT1 | CPT2 | CPT2_HUMAN | Carnitine O-palmitoyltransferase 2, mitochondrial | Carnitine palmitoyltransferase 2 | Carnitine palmitoyltransferase II |
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| Type: | PROTEIN |
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| Mol. Mass.: | 73789.25 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_887455 |
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| Residue: | 658 |
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| Sequence: | MVPRLLLRAWPRGPAVGPGAPSRPLSAGSGPGQYLQRSIVPTMHYQDSLPRLPIPKLEDT
IRRYLSAQKPLLNDGQFRKTEQFCKSFENGIGKELHEQLVALDKQNKHTSYISGPWFDMY
LSARDSVVLNFNPFMAFNPDPKSEYNDQLTRATNMTVSAIRFLKTLRAGLLEPEVFHLNP
AKSDTITFKRLIRFVPSSLSWYGAYLVNAYPLDMSQYFRLFNSTRLPKPSRDELFTDDKA
RHLLVLRKGNFYIFDVLDQDGNIVSPSEIQAHLKYILSDSSPAPEFPLAYLTSENRDIWA
ELRQKLMSSGNEESLRKVDSAVFCLCLDDFPIKDLVHLSHNMLHGDGTNRWFDKSFNLII
AKDGSTAVHFEHSWGDGVAVLRFFNEVFKDSTQTPAVTPQSQPATTDSTVTVQKLNFELT
DALKTGITAAKEKFDATMKTLTIDCVQFQRGGKEFLKKQKLSPDAVAQLAFQMAFLRQYG
QTVATYESCSTAAFKHGRTETIRPASVYTKRCSEAFVREPSRHSAGELQQMMVECSKYHG
QLTKEAAMGQGFDRHLFALRHLAAAKGIILPELYLDPAYGQINHNVLSTSTLSSPAVNLG
GFAPVVSDGFGVGYAVHDNWIGCNVSSYPGRNAREFLQCVEKALEDMFDALEGKSIKS
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| BDBM50403031 |
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| n/a |
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| Name | BDBM50403031 |
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| Synonyms: | CHEMBL2216771 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H14O5S |
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| Mol. Mass. | 342.366 |
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| SMILES | OC(=O)C(=O)c1ccc(OCCOc2ccc3ccccc3c2)s1 |
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| Structure | 
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