| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Thromboxane A2 receptor |
|---|
| Ligand | BDBM50003795 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_209756 (CHEMBL815547) |
|---|
| Kd | 1258.93±n/a nM |
|---|
| Citation |  Campbell, I; Collington, E; Finch, H; Hayes, R; Lumley, P; Mills, K; Robertson, G; Wharton, K; Watts, I Synthesis and pharmacological evaluation of combined Thromboxane receptor antagonists/thromboxane synthase inhibitors: Pyridine-containing amino-prostanoids Bioorg Med Chem Lett1:695-698 (1991) Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Thromboxane A2 receptor |
|---|
| Name: | Thromboxane A2 receptor |
|---|
| Synonyms: | TA2R_RAT | TXA2/PGH2 | Tbxa2r | Thromboxane A2 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 36943.05 |
|---|
| Organism: | RAT |
|---|
| Description: | Thromboxane A2 TBXA2R RAT::P34978 |
|---|
| Residue: | 341 |
|---|
| Sequence: | MWLNSTSLGACFRPVNITLQERRAIASPWFAASFCALGLGSNLLALSVLAGARPGAGPRS
SFLALLCGLVLTDFLGLLVTGAVVASQHAALLDWRATDPGCRLCHFMGAAMVFFGLCPLL
LGAAMAAERFVGITRPFSRPAATSRRAWATVGLVWVGAGTLGLLPLLGLGRYSVQYPGSW
CFLTLGAERGDVAFGLMFALLGSVSVGLSLLLNTVSVATLCRVYHAREATQRPRDCEVEM
MVQLVGIMVVATVCWMPLLVFILQTLLQTLPVMSPSGQLLRTTERQLLIYLRVATWNQIL
DPWVYILFRRSVLRRLHPRFTSQLQAVSLHSPPTQAMLSGP
|
|
|
|---|
| BDBM50003795 |
|---|
| n/a |
|---|
| Name | BDBM50003795 |
|---|
| Synonyms: | 5-[1-Pyridin-3-yl-1-(3-trifluoromethyl-phenyl)-meth-(E)-ylideneaminooxy]-pentanoic acid | 5-[Pyridin-3-yl-(3-trifluoromethyl-phenyl)-methyleneaminooxy]-pentanoic acid | CHEMBL280728 | R-68070 | ridogrel |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C18H17F3N2O3 |
|---|
| Mol. Mass. | 366.3344 |
|---|
| SMILES | OC(=O)CCCCO\N=C(\c1cccnc1)c1cccc(c1)C(F)(F)F |
|---|
| Structure | 
|
|---|
Search and Browse
