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TargetHydroxyacid oxidase 1
LigandBDBM50404998
Substrate/Competitorn/a
Meas. Tech.ChEMBL_71275
IC50 180±n/a nM
Citation Williams HWEichler ERandall WCRooney CSCragoe EJStreeter KBSchwam HMichelson SRPatchett AATaub D Inhibitors of glycolic acid oxidase. 4-substituted 2,4-dioxobutanoic acid derivatives. J Med Chem 26:1196-200 (1983) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Hydroxyacid oxidase 1
Name:Hydroxyacid oxidase 1
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:40927.89
Organism:Homo sapiens (Human)
Description:ChEMBL_71275
Residue:370
Sequence:
MLPRLICINDYEQHAKSVLPKSIYDYYRSGANDEETLADNIAAFSRWKLYPRMLRNVAET
DLSTSVLGQRVSMPICVGATAMQRMAHVDGELATVRACQSLGTGMMLSSWATSSIEEVAE
AGPEALRWLQLYIYKDREVTKKLVRQAEKMGYKAIFVTVDTPYLGNRLDDVRNRFKLPPQ
LRMKNFETSTLSFSPEENFGDDSGLAAYVAKAIDPSISWEDIKWLRRLTSLPIVAKGILR
GDDAREAVKHGLNGILVSNHGARQLDGVPATIDVLPEIVEAVEGKVEVFLDGGVRKGTDV
LKALALGAKAVFVGRPIVWGLAFQGEKGVQDVLEILKEEFRLAMALSGCQNVKVIDKTLV
RKNPLAVSKI
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  Blast E-value cutoff:
BDBM50404998
n/a
NameBDBM50404998
Synonyms:CHEMBL276330
TypeSmall organic molecule
Emp. Form.C24H17NO4
Mol. Mass.383.3961
SMILESOC(=O)C(=O)CC(=O)c1ccc(cc1)-n1c(cc2ccccc12)-c1ccccc1
Structure
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