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TargetSerotonin 1d (5-HT1d) receptor
LigandBDBM50406771
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1958
IC50 0.316±n/a nM
Citation Street LJBaker RDavey WBGuiblin ARJelley RAReeve AJRoutledge HSternfeld FWatt APBeer MS Synthesis and serotonergic activity of N,N-dimethyl-2-[5-(1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]ethylamine and analogues: potent agonists for 5-HT1D receptors. J Med Chem 38:1799-810 (1995) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Serotonin 1d (5-HT1d) receptor
Name:Serotonin 1d (5-HT1d) receptor
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:32680.56
Organism:Sus scrofa
Description:ChEMBL_1963
Residue:291
Sequence:
AMTDLLVSILVMPISIPYTITQTWSFGQLLCDIWLSSDITCCTASILHLCVIALDRYWAI
TDALEYSKRRTAGHAAAMIAIVWAISICISIPPLFWRQARAHEEISDCLVNTSQISYTIY
STCGAFYIPSLLLIILYGRIYRAARNRILNPPSLYGKRFTTAHLITGSAGSSLCSLNPSL
HEGHSHSAGSPLFFNHVKIKLADSVLERKRISAARERKATKTLGIILGAFIICWLPFFVA
SLVLPICRDSCWIHPALFDFFTWLGYLNSLINPIIYTVFNEEFRQAFQKVV
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  Blast E-value cutoff:
BDBM50406771
n/a
NameBDBM50406771
Synonyms:L-694247
TypeSmall organic molecule
Emp. Form.C20H21N5O3S
Mol. Mass.411.477
SMILESCS(=O)(=O)Nc1ccc(Cc2noc(n2)-c2ccc3[nH]cc(CCN)c3c2)cc1
Structure
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