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TargetPeptide deformylase
LigandBDBM50416428
Substrate/Competitorn/a
Meas. Tech.ChEMBL_643979 (CHEMBL1211878)
IC50 28±n/a nM
Citation Lee, SKChoi, KHLee, SJSuh, SWKim, BMLee, BJ Peptide deformylase inhibitors with retro-amide scaffold: synthesis and structure-activity relationships. Bioorg Med Chem Lett20:4317-9 (2010) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Peptide deformylase
Name:Peptide deformylase
Synonyms:DEF_PSEAE | PDF | Polypeptide deformylase | def
Type:PROTEIN
Mol. Mass.:19357.88
Organism:Pseudomonas aeruginosa
Description:ChEMBL_643979
Residue:168
Sequence:
MAILNILEFPDPRLRTIAKPVEVVDDAVRQLIDDMFETMYEAPGIGLAATQVNVHKRIVV
MDLSEDKSEPRVFINPEFEPLTEDMDQYQEGCLSVPGFYENVDRPQKVRIKALDRDGNPF
EEVAEGLLAVCIQHECDHLNGKLFVDYLSTLKRDRIRKKLEKQHRQQA
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50416428
n/a
NameBDBM50416428
Synonyms:CHEMBL1209044
TypeSmall organic molecule
Emp. Form.C19H34N4O5
Mol. Mass.398.4971
SMILESCC(C)(C)[C@H](NC(=O)N1CCOCC1)C(=O)N(CC1CCCC1)CC(=O)NO |r|
Structure
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