| Reaction Details |
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 | Report a problem with these data |
| Target | Solute carrier family 22 member 8 |
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| Ligand | BDBM50390999 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_838512 (CHEMBL2078140) |
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| Ki | 1890±n/a nM |
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| Citation |  Takeda, M; Babu, E; Narikawa, S; Endou, H Interaction of human organic anion transporters with various cephalosporin antibiotics. Eur J Pharmacol438:137-42 (2002) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Solute carrier family 22 member 8 |
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| Name: | Solute carrier family 22 member 8 |
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| Synonyms: | OAT3 | Organic anion transporter 3 | S22A8_HUMAN | SLC22A8 | hOAT3 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 59870.13 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1486920 |
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| Residue: | 542 |
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| Sequence: | MTFSEILDRVGSMGHFQFLHVAILGLPILNMANHNLLQIFTAATPVHHCRPPHNASTGPW
VLPMGPNGKPERCLRFVHPPNASLPNDTQRAMEPCLDGWVYNSTKDSIVTEWDLVCNSNK
LKEMAQSIFMAGILIGGLVLGDLSDRFGRRPILTCSYLLLAASGSGAAFSPTFPIYMVFR
FLCGFGISGITLSTVILNVEWVPTRMRAIMSTALGYCYTFGQFILPGLAYAIPQWRWLQL
TVSIPFFVFFLSSWWTPESIRWLVLSGKSSKALKILRRVAVFNGKKEEGERLSLEELKLN
LQKEISLAKAKYTASDLFRIPMLRRMTFCLSLAWFATGFAYYSLAMGVEEFGVNLYILQI
IFGGVDVPAKFITILSLSYLGRHTTQAAALLLAGGAILALTFVPLDLQTVRTVLAVFGKG
CLSSSFSCLFLYTSELYPTVIRQTGMGVSNLWTRVGSMVSPLVKITGEVQPFIPNIIYGI
TALLGGSAALFLPETLNQPLPETIEDLENWSLRAKKPKQEPEVEKASQRIPLQPHGPGLG
SS
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| BDBM50390999 |
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| n/a |
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| Name | BDBM50390999 |
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| Synonyms: | CEFOPERAZONE |
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| Type | Small organic molecule |
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| Emp. Form. | C25H27N9O8S2 |
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| Mol. Mass. | 645.667 |
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| SMILES | CCN1CCN(C(=O)N[C@@H](C(=O)N[C@H]2[C@H]3SCC(CSc4nnnn4C)=C(N3C2=O)C(O)=O)c2ccc(O)cc2)C(=O)C1=O |c:26| |
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| Structure | 
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