Ki Summary

Reaction Details

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Target

Solute carrier family 15 member 2

Ligand

BDBM50370592

Substrate/Competitor

n/a

Meas. Tech.

ChEMBL_838253 (CHEMBL2076201)

>10000000±n/a nM

Citation

Luckner, P; Brandsch, M Interaction of 31 beta-lactam antibiotics with the H+/peptide symporter PEPT2: analysis of affinity constants and comparison with PEPT1. Eur J Pharm Biopharm59:17-24 (2004) [PubMed] Article

More Info.:

Get all data from this article, Assay Method

Solute carrier family 15 member 2

Name:

Solute carrier family 15 member 2

Synonyms:

Oligopeptide transporter, kidney isoform | Pept2 | S15A2_RAT | Slc15a2

Type:

PROTEIN

Mol. Mass.:

81331.63

Organism:

Rattus norvegicus

Description:

ChEMBL_838253

Residue:

729

Sequence:

MNPFQKNESKETLFSPVSTEEMLPRPPSPPKKSPPKIFGSSYPVSIAFIVVNEFCERFSY
YGMKAVLTLYFLYFLHWNEDTSTSVYHAFSSLCYFTPILGAAIADSWLGKFKTIIYLSLV
YVLGHVFKSLGAIPILGGKMLHTILSLVGLSLIALGTGGIKPCVAAFGGDQFEEEHAEAR
TRYFSVFYLAINAGSLISTFITPMLRGDVKCFGQDCYALAFGVPGLLMVLALVVFAMGSK
MYRKPPPEGNIVAQVIKCIWFALCNRFRNRSGDLPKRQHWLDWAAEKYPKHLIADVKALT
RVLFLYIPLPMFWALLDQQGSRWTLQANKMNGDLGFFVLQPDQMQVLNPFLVLIFIPLFD
LVIYRLISKCRINFSSLRKMAVGMILACLAFAVAALVETKINGMIHPQPASQEIFLQVLN
LADGDVKVTVLGSRNNSLLVESVSSFQNTTHYSKLHLEAKSQDLHFHLKYNSLSVHNDHS
VEEKNCYQLLIHQDGESISSMLVKDTGIKPANGMAAIRFINTLHKDLNISLDTDAPLSVG
KDYGVSAYRTVLRGKYPAVHCETEDKVFSLDLGQLDFGTTYLFVITNITSQGLQAWKAED
IPVNKLSIAWQLPQYVLVTAAEVMFSVTGLEFSYSQAPSSMKSVLQAAWLLTVAVGNIIV
LVVAQFSGLAQWAEFVLFSCLLLVVCLIFSVMAYYYVPLKSEDTREATDKQIPAVQGNMI
NLETKNTRL

BDBM50370592

n/a

Name

BDBM50370592

Synonyms:

CEPHAPIRIN | Cefa-Lak | Cefadyl | Cefapirin

Type

Small organic molecule

Emp. Form.

C17H17N3O6S2

Mol. Mass.

423.463

SMILES

CC(=O)OCC1=C(N2[C@H](SC1)[C@H](NC(=O)CSc1ccncc1)C2=O)C(O)=O |r,t:5|

Structure