| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 1 |
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| Ligand | BDBM50423303 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_456079 (CHEMBL888088) |
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| Kd | 1.2±n/a nM |
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| Citation |  Troxler, T; Hoyer, D; Langenegger, D; Neumann, P; Pfäffli, P; Schoeffter, P; Sorg, D; Swoboda, R; Hurth, K Identification and SAR of potent and selective non-peptide obeline somatostatin sst1 receptor antagonists. Bioorg Med Chem Lett17:3983-7 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 1 |
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| Name: | Somatostatin receptor type 1 |
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| Synonyms: | SOMATOSTATIN SST1 | SRIF-2 | SS1R | SSR1_RAT | Somatostatin receptor | Somatostatin receptor type 1 | Sstr1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 42752.93 |
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| Organism: | RAT |
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| Description: | SOMATOSTATIN SST1 SSTR1 RAT::P28646 |
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| Residue: | 391 |
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| Sequence: | MFPNGTAPSPTSSPSSSPGGCGEGVCSRGPGSGAADGMEEPGRNSSQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCASRISTL
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| BDBM50423303 |
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| n/a |
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| Name | BDBM50423303 |
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| Synonyms: | CHEMBL248907 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H29BrN6O2S |
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| Mol. Mass. | 557.506 |
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| SMILES | COc1ccc(Br)c2C[C@@H]3[C@H](C[C@H](CN3C)C(=O)N3CCN(CC3)c3ccc4nsnc4n3)Cc12 |
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| Structure | 
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