| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 2 |
|---|
| Ligand | BDBM50423310 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_456080 (CHEMBL888089) |
|---|
| Kd | 7762±n/a nM |
|---|
| Citation |  Troxler, T; Hoyer, D; Langenegger, D; Neumann, P; Pfäffli, P; Schoeffter, P; Sorg, D; Swoboda, R; Hurth, K Identification and SAR of potent and selective non-peptide obeline somatostatin sst1 receptor antagonists. Bioorg Med Chem Lett17:3983-7 (2007) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Somatostatin receptor type 2 |
|---|
| Name: | Somatostatin receptor type 2 |
|---|
| Synonyms: | SOMATOSTATIN SST2 | SRIF-1 | SS2R | SSR2_RAT | Somatostatin receptor | Somatostatin receptor 2 | Somatostatin receptor type 2 | Sstr2 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 41212.21 |
|---|
| Organism: | RAT |
|---|
| Description: | SOMATOSTATIN SST2 SSTR2 RAT::P30680 |
|---|
| Residue: | 369 |
|---|
| Sequence: | MELTSEQFNGSQVWIPSPFDLNGSLGPSNGSNQTEPYYDMTSNAVLTFIYFVVCVVGLCG
NTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMT
VDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMINVAVWGVSLLVILPIMIY
AGLRSNQWGRSSCTINWPGESGAWYTGFIIYAFILGFLVPLTIICLCYLFIIIKVKSSGI
RVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSVAISPTPALKGMFDFVVIL
TYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGAEDGERSDSKQDKSRLNETTETQRTL
LNGDLQTSI
|
|
|
|---|
| BDBM50423310 |
|---|
| n/a |
|---|
| Name | BDBM50423310 |
|---|
| Synonyms: | CHEMBL251543 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C25H30N4O4 |
|---|
| Mol. Mass. | 450.5301 |
|---|
| SMILES | CN1C[C@@H](C[C@@H]2Cc3c(O)cccc3C[C@@H]12)C(=O)N1CCN(CC1)c1ccc(cc1)[N+]([O-])=O |
|---|
| Structure | 
|
|---|
Search and Browse
