| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 2 |
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| Ligand | BDBM50423484 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_461986 (CHEMBL944829) |
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| Kd | 5888±n/a nM |
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| Citation |  Troxler, T; Enz, A; Hoyer, D; Langenegger, D; Neumann, P; Pfäffli, P; Schoeffter, P; Hurth, K Ergoline derivatives as highly potent and selective antagonists at the somatostatin sst 1 receptor. Bioorg Med Chem Lett18:979-82 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 2 |
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| Name: | Somatostatin receptor type 2 |
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| Synonyms: | SOMATOSTATIN SST2 | SRIF-1 | SS2R | SSR2_RAT | Somatostatin receptor | Somatostatin receptor 2 | Somatostatin receptor type 2 | Sstr2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 41212.21 |
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| Organism: | RAT |
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| Description: | SOMATOSTATIN SST2 SSTR2 RAT::P30680 |
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| Residue: | 369 |
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| Sequence: | MELTSEQFNGSQVWIPSPFDLNGSLGPSNGSNQTEPYYDMTSNAVLTFIYFVVCVVGLCG
NTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMT
VDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMINVAVWGVSLLVILPIMIY
AGLRSNQWGRSSCTINWPGESGAWYTGFIIYAFILGFLVPLTIICLCYLFIIIKVKSSGI
RVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSVAISPTPALKGMFDFVVIL
TYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGAEDGERSDSKQDKSRLNETTETQRTL
LNGDLQTSI
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| BDBM50423484 |
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| n/a |
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| Name | BDBM50423484 |
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| Synonyms: | CHEMBL401131 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H28Cl2N4O |
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| Mol. Mass. | 483.433 |
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| SMILES | CN1C[C@@H](C[C@H]2[C@H]1Cc1c(Cl)[nH]c3cccc2c13)C(=O)N1CCN(CC1)c1ccc(Cl)cc1 |
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| Structure | 
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