| Reaction Details |
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 | Report a problem with these data |
| Target | Acetylpolyamine amidohydrolase (APAH) |
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| Ligand | BDBM50438390 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_975718 |
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| IC50 | 270±n/a nM |
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| Citation |  Decroos C; Bowman CM; Christianson DW Synthesis and evaluation of N8-acetylspermidine analogues as inhibitors of bacterial acetylpolyamine amidohydrolase. Bioorg Med Chem 21:4530-40 (2013) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Acetylpolyamine amidohydrolase (APAH) |
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| Name: | Acetylpolyamine amidohydrolase (APAH) |
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| Synonyms: | Acetylpolyamine aminohydrolase |
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| Type: | Protein |
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| Mol. Mass.: | 36324.64 |
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| Organism: | Mycoplana ramosa (Gram-negative bacterium) |
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| Description: | n/a |
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| Residue: | 341 |
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| Sequence: | MRVIFSEDHKLRNAKTELYGGELVPPFEAPFRAEWILAAVKEAGFDDVVAPARHGLETVL
KVHDAGYLNFLETAWDRWKAAGYKGEAIATSFPVRRTSPRIPTDIEGQIGYYCNAAETAI
SPGTWEAALSSMASAIDGADLIAAGHKAAFSLCRPPGHHAGIDMFGGYCFINNAAVAAQR
LLDKGAKKIAILDVDFHHGNGTQDIFYERGDVFFASLHGDPAEAFPHFLGYAEETGKGAG
AGTTANYPMGRGTPYSVWGEALTDSLKRIAAFGAEAIVVSLGVDTFEQDPISFFKLTSPD
YITMGRTIAASGVPLLVVMEGGYGVPEIGLNVANVLKGVAG
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| BDBM50438390 |
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| n/a |
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| Name | BDBM50438390 |
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| Synonyms: | CHEMBL2414000 |
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| Type | Small organic molecule |
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| Emp. Form. | C10H19F3N2O |
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| Mol. Mass. | 240.2659 |
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| SMILES | NCCCNCCCCCC(=O)C(F)(F)F |
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| Structure | 
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