| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Vasoactive intestinal polypeptide receptor 2 |
|---|
| Ligand | BDBM50445109 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_1284427 (CHEMBL3106155) |
|---|
| EC50 | 0.21±n/a nM |
|---|
| Citation |  Giordanetto, F; Revell, JD; Knerr, L; Hostettler, M; Paunovic, A; Priest, C; Janefeldt, A; Gill, A Stapled Vasoactive Intestinal Peptide (VIP) Derivatives Improve VPAC2 Agonism and Glucose-Dependent Insulin Secretion. ACS Med Chem Lett4:1163-8 (2013) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Vasoactive intestinal polypeptide receptor 2 |
|---|
| Name: | Vasoactive intestinal polypeptide receptor 2 |
|---|
| Synonyms: | VIP 2 | VIP2R | VIPR2 | VIPR2_HUMAN |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 49488.30 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | VIP 2 VIPR2 HUMAN::P41587 |
|---|
| Residue: | 438 |
|---|
| Sequence: | MRTLLPPALLTCWLLAPVNSIHPECRFHLEIQEEETKCAELLRSQTEKHKACSGVWDNIT
CWRPANVGETVTVPCPKVFSNFYSKAGNISKNCTSDGWSETFPDFVDACGYSDPEDESKI
TFYILVKAIYTLGYSVSLMSLATGSIILCLFRKLHCTRNYIHLNLFLSFILRAISVLVKD
DVLYSSSGTLHCPDQPSSWVGCKLSLVFLQYCIMANFFWLLVEGLYLHTLLVAMLPPRRC
FLAYLLIGWGLPTVCIGAWTAARLYLEDTGCWDTNDHSVPWWVIRIPILISIIVNFVLFI
SIIRILLQKLTSPDVGGNDQSQYKRLAKSTLLLIPLFGVHYMVFAVFPISISSKYQILFE
LCLGSFQGLVVAVLYCFLNSEVQCELKRKWRSRCPTPSASRDYRVCGSSFSRNGSEGALQ
FHRGSRAQSFLQTETSVI
|
|
|
|---|
| BDBM50445109 |
|---|
| n/a |
|---|
| Name | BDBM50445109 |
|---|
| Synonyms: | CHEMBL3102922 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C158H256N46O46 |
|---|
| Mol. Mass. | 3536.0038 |
|---|
| SMILES | n/a |
|---|
| Structure | 
|
|---|
Search and Browse
