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TargetNeuropeptide Y receptor type 2
LigandBDBM50445636
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1284012 (CHEMBL3107076)
IC50 25±n/a nM
Citation Mittapalli, GKRoberts, E Ligands of the neuropeptide Y Y2 receptor. Bioorg Med Chem Lett24:430-41 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Neuropeptide Y receptor type 2
Name:Neuropeptide Y receptor type 2
Synonyms:NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:Enzyme Catalytic Domain
Mol. Mass.:42734.65
Organism:Homo sapiens (Human)
Description:NPY-Y2 NPY2R HUMAN::P49146
Residue:381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSI
ILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGP
VLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLA
SPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYT
RIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDL
KEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAK
KNLEVRKNSGPNDSFTEATNV
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50445636
n/a
NameBDBM50445636
Synonyms:CHEMBL3104201
TypeSmall organic molecule
Emp. Form.C28H36FN3O3
Mol. Mass.481.6021
SMILESCCN(CC)C(=O)C(C1CCN(CC1)c1ccc(NC(=O)C2CCOC2)cc1F)c1ccccc1
Structure
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