| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A3 |
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| Ligand | BDBM50051336 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_30324 (CHEMBL638578) |
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| Ki | 741±n/a nM |
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| Citation |  Moro, S; van Rhee, AM; Sanders, LH; Jacobson, KA Flavonoid derivatives as adenosine receptor antagonists: a comparison of the hypothetical receptor binding site based on a comparative molecular field analysis model. J Med Chem41:46-52 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A3 |
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| Name: | Adenosine receptor A3 |
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| Synonyms: | A3 adenosine receptor (hA3) | AA3R_HUMAN | ADORA3 | Adenosine A3 receptor (A3AR) |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 36197.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P0DMS8 |
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| Residue: | 318 |
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| Sequence: | MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIA
VGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKR
VTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYF
SFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFA
LSWLPLSIINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKAC
VVCHPSDSLDTSIEKNSE
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| BDBM50051336 |
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| n/a |
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| Name | BDBM50051336 |
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| Synonyms: | 3,7-Diethoxy-5-hydroxy-2-phenyl-chromen-4-one | CHEMBL449090 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H18O5 |
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| Mol. Mass. | 326.3432 |
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| SMILES | CCOc1cc(O)c2c(c1)oc(-c1ccccc1)c(OCC)c2=O |
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| Structure | 
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