| Reaction Details |
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 | Report a problem with these data |
| Target | Cytohesin-3 |
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| Ligand | BDBM50013327 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1348972 (CHEMBL3265619) |
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| IC50 | 38000±n/a nM |
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| Citation |  Kim, Y; Yoon, Y Elucidation of different inhibition mechanism of small chemicals on PtdInsP-binding domains using in silico docking experiments. Bioorg Med Chem Lett24:2256-62 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cytohesin-3 |
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| Name: | Cytohesin-3 |
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| Synonyms: | ARNO3 | CYH3_HUMAN | CYTH3 | GRP1 | General receptor of phosphoinositides 1 (GRP1) | PSCD3 |
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| Type: | Enzyme |
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| Mol. Mass.: | 46340.05 |
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| Organism: | Homo sapiens (Human) |
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| Description: | O43739 |
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| Residue: | 400 |
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| Sequence: | MDEDGGGEGGGVPEDLSLEEREELLDIRRRKKELIDDIERLKYEIAEVMTEIDNLTSVEE
SKTTQRNKQIAMGRKKFNMDPKKGIQFLIENDLLQSSPEDVAQFLYKGEGLNKTVIGDYL
GERDEFNIKVLQAFVELHEFADLNLVQALRQFLWSFRLPGEAQKIDRMMEAFASRYCLCN
PGVFQSTDTCYVLSFAIIMLNTSLHNHNVRDKPTAERFIAMNRGINEGGDLPEELLRNLY
ESIKNEPFKIPEDDGNDLTHTFFNPDREGWLLKLGGGRVKTWKRRWFILTDNCLYYFEYT
TDKEPRGIIPLENLSIREVEDPRKPNCFELYNPSHKGQVIKACKTEADGRVVEGNHVVYR
ISAPSPEEKEEWMKSIKASISRDPFYDMLATRKRRIANKK
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| BDBM50013327 |
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| n/a |
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| Name | BDBM50013327 |
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| Synonyms: | CHEMBL3263343 |
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| Type | Small organic molecule |
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| Emp. Form. | C4H5N2O5P |
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| Mol. Mass. | 192.0667 |
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| SMILES | OC(=O)c1cc(n[nH]1)P(O)(O)=O |
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| Structure | 
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