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TargetD-alanyl-D-alanine dipeptidase
LigandBDBM50014158
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1350288 (CHEMBL3267626)
Ki 6100±n/a nM
Citation Muthyala, RRastogi, NShin, WSPeterson, MLSham, YY Cell permeable vanX inhibitors as vancomycin re-sensitizing agents. Bioorg Med Chem Lett24:2535-8 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
D-alanyl-D-alanine dipeptidase
Name:D-alanyl-D-alanine dipeptidase
Synonyms:D-Ala-D-Ala dipeptidase | VANX_ENTFC | Vancomycin B-type resistance protein vanX | vanX
Type:PROTEIN
Mol. Mass.:23377.40
Organism:Enterococcus faecium
Description:ChEMBL_1350288
Residue:202
Sequence:
MEIGFTFLDEIVHGVRWDAKYATWDNFTGKPVDGYEVNRIVGTYELAESLLKAKELAATQ
GYGLLLWDGYRPKRAVNCFMQWAAQPENNLTKESYYPNIDRTEMISKGYVASKSSHSRGS
AIDLTLYRLDTGELVPMGSRFDFMDERSHHAANGISCNEAQNRRRLRSIMENSGFEAYSL
EWWHYVLRDEPYPNSYFDFPVK
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  Blast E-value cutoff:
BDBM50014158
n/a
NameBDBM50014158
Synonyms:CHEMBL3260856
TypeSmall organic molecule
Emp. Form.C8H18NO4P
Mol. Mass.223.2066
SMILESCC(C)[C@H](CP(O)(=O)[C@@H](C)N)C(O)=O |r|
Structure
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