| Reaction Details |
|---|
 | Report a problem with these data |
| Target | 4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9 |
|---|
| Ligand | BDBM92459 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_1432745 (CHEMBL3390549) |
|---|
| IC50 | 59000±n/a nM |
|---|
| Citation |  Seelhorst, K; Piernitzki, T; Lunau, N; Meier, C; Hahn, U Synthesis and analysis of potentiala1,3-fucosyltransferase inhibitors. Bioorg Med Chem22:6430-7 (2014) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| 4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9 |
|---|
| Name: | 4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9 |
|---|
| Synonyms: | Alpha-(1,3)-fucosyltransferase 9 | FUT9 | FUT9_HUMAN | Fuc-TIX | FucT-IX | Fucosyltransferase 9 | Fucosyltransferase IX | Galactoside 3-L-fucosyltransferase |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 42078.14 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_10775 |
|---|
| Residue: | 359 |
|---|
| Sequence: | MTSTSKGILRPFLIVCIILGCFMACLLIYIKPTNSWIFSPMESASSVLKMKNFFSTKTDY
FNETTILVWVWPFGQTFDLTSCQAMFNIQGCHLTTDRSLYNKSHAVLIHHRDISWDLTNL
PQQARPPFQKWIWMNLESPTHTPQKSGIEHLFNLTLTYRRDSDIQVPYGFLTVSTNPFVF
EVPSKEKLVCWVVSNWNPEHARVKYYNELSKSIEIHTYGQAFGEYVNDKNLIPTISTCKF
YLSFENSIHKDYITEKLYNAFLAGSVPVVLGPSRENYENYIPADSFIHVEDYNSPSELAK
YLKEVDKNNKLYLSYFNWRKDFTVNLPRFWESHACLACDHVKRHQEYKSVGNLEKWFWN
|
|
|
|---|
| BDBM92459 |
|---|
| n/a |
|---|
| Name | BDBM92459 |
|---|
| Synonyms: | CHEMBL384759 | GDP | Guanosine Diphosphate |
|---|
| Type | Small molecule |
|---|
| Emp. Form. | C10H15N5O11P2 |
|---|
| Mol. Mass. | 443.2005 |
|---|
| SMILES | Nc1nc2n(cnc2c(=O)[nH]1)[C@@H]1O[C@H](COP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]1O |
|---|
| Structure | 
|
|---|
Search and Browse
