| Reaction Details |
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 | Report a problem with these data |
| Target | Glutathione S-transferase P |
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| Ligand | BDBM50038321 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1441152 (CHEMBL3378816) |
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| IC50 | 500±n/a nM |
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| Citation |  Rotili, D; De Luca, A; Tarantino, D; Pezzola, S; Forgione, M; Morozzo Della Rocca, B; Falconi, M; Mai, A; Caccuri, AM Synthesis and structure--activity relationship of new cytotoxic agents targeting human glutathione-S-transferases. Eur J Med Chem89:156-71 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Glutathione S-transferase P |
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| Name: | Glutathione S-transferase P |
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| Synonyms: | FAEES3 | GST class-pi | GST3 | GSTP1 | GSTP1-1 | GSTP1_HUMAN | Glutathione S-transferase | Glutathione S-transferase (GST) | Glutathione S-transferase P | Glutathione S-transferase Pi | Glutathione transferase (GST) |
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| Type: | Enzyme |
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| Mol. Mass.: | 23353.53 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P09211 |
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| Residue: | 210 |
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| Sequence: | MPPYTVVYFPVRGRCAALRMLLADQGQSWKEEVVTVETWQEGSLKASCLYGQLPKFQDGD
LTLYQSNTILRHLGRTLGLYGKDQQEAALVDMVNDGVEDLRCKYISLIYTNYEAGKDDYV
KALPGQLKPFETLLSQNQGGKTFIVGDQISFADYNLLDLLLIHEVLAPGCLDAFPLLSAY
VGRLSARPKLKAFLASPEYVNLPINGNGKQ
|
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|
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| BDBM50038321 |
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| n/a |
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| Name | BDBM50038321 |
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| Synonyms: | CHEMBL3360505 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H13N3O3S |
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| Mol. Mass. | 315.347 |
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| SMILES | [O-][N+](=O)c1ccc(SCCCc2ccccc2)c2nonc12 |
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| Structure | 
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