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TargetLipoxygenase
LigandBDBM50021468
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1457228 (CHEMBL3370272)
IC50 29280±n/a nM
Citation Bukhari, SNLauro, GJantan, IBifulco, GAmjad, MW Pharmacological evaluation and docking studies ofa,ß-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines. Bioorg Med Chem22:4151-61 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Lipoxygenase
Name:Lipoxygenase
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:1886.07
Organism:Glycine max
Description:ChEMBL_103841
Residue:18
Sequence:
PNSEEGLTCRGIPNSISI
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BDBM50021468
n/a
NameBDBM50021468
Synonyms:CHEMBL3289934
TypeSmall organic molecule
Emp. Form.C24H26N4O5
Mol. Mass.450.487
SMILESCN(C)c1ccc(\C=C2\CCC\C(=C/c3ccc(cc3[N+]([O-])=O)N(C)C)C2=O)c(c1)[N+]([O-])=O
Structure
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