| Reaction Details |
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 | Report a problem with these data |
| Target | Protein tyrosine phosphatase type IVA 1 |
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| Ligand | BDBM50059139 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1461024 (CHEMBL3395082) |
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| IC50 | 209000±n/a nM |
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| Citation |  Hoeger, B; Diether, M; Ballester, PJ; Köhn, M Biochemical evaluation of virtual screening methods reveals a cell-active inhibitor of the cancer-promoting phosphatases of regenerating liver. Eur J Med Chem88:89-100 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Protein tyrosine phosphatase type IVA 1 |
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| Name: | Protein tyrosine phosphatase type IVA 1 |
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| Synonyms: | PRL1 | PTP4A1 | PTPCAAX1 | TP4A1_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 19823.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1461024 |
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| Residue: | 173 |
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| Sequence: | MARMNRPAPVEVTYKNMRFLITHNPTNATLNKFIEELKKYGVTTIVRVCEATYDTTLVEK
EGIHVLDWPFDDGAPPSNQIVDDWLSLVKIKFREEPGCCIAVHCVAGLGRAPVLVALALI
EGGMKYEDAVQFIRQKRRGAFNSKQLLYLEKYRPKMRLRFKDSNGHRNNCCIQ
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| BDBM50059139 |
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| n/a |
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| Name | BDBM50059139 |
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| Synonyms: | CHEMBL3393147 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H9NO3S |
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| Mol. Mass. | 271.291 |
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| SMILES | OC(=O)c1ccc[n+]2c([O-])c(sc12)-c1ccccc1 |
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| Structure | 
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