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TargetSimilar to alpha-tubulin isoform 1
LigandBDBM50086309
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1475978 (CHEMBL3428203)
IC50 7890±n/a nM
Citation Qin, YJLi, YJJiang, AQYang, MRZhu, QZDong, HZhu, HL Design, synthesis and biological evaluation of novel pyrazoline-containing derivatives as potential tubulin assembling inhibitors. Eur J Med Chem94:447-57 (2015) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Similar to alpha-tubulin isoform 1
Name:Similar to alpha-tubulin isoform 1
Synonyms:Similar to alpha-tubulin isoform 1
Type:PROTEIN
Mol. Mass.:10383.05
Organism:Bos taurus
Description:ChEMBL_104716
Residue:99
Sequence:
CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGK
HVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50086309
n/a
NameBDBM50086309
Synonyms:CHEMBL3426003
TypeSmall organic molecule
Emp. Form.C26H23FN2O6
Mol. Mass.478.469
SMILESCOc1cc(cc(OC)c1OC)C(=O)N1N=C(CC1c1ccc2OCOc2c1)c1ccc(F)cc1 |c:16|
Structure
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