| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Long-chain fatty acid transport protein 2 |
|---|
| Ligand | BDBM50168142 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_1576582 (CHEMBL3807377) |
|---|
| IC50 | 6300±n/a nM |
|---|
| Citation |  Black, PN; Ahowesso, C; Montefusco, D; Saini, N; DiRusso, CC Fatty Acid Transport Proteins: Targeting FATP2 as a Gatekeeper Involved in the Transport of Exogenous Fatty Acids. Medchemcomm7:612-622 (2016) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Long-chain fatty acid transport protein 2 |
|---|
| Name: | Long-chain fatty acid transport protein 2 |
|---|
| Synonyms: | 6.2.1.- | 6.2.1.3 | ACSVL1 | ACSVL1 | FACVL1 | FATP-2 | FATP2 | Fatty acid transport protein 2 | Fatty-acid-coenzyme A ligase, very long-chain 1 | Long-chain-fatty-acid--CoA ligase | S27A2_HUMAN | SLC27A2 | Solute carrier family 27 member 2 | THCA-CoA ligase | VLACS | Very long-chain acyl-CoA synthetase |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 70329.11 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_100784 |
|---|
| Residue: | 620 |
|---|
| Sequence: | MLSAIYTVLAGLLFLPLLVNLCCPYFFQDIGYFLKVAAVGRRVRSYGKRRPARTILRAFL
EKARQTPHKPFLLFRDETLTYAQVDRRSNQVARALHDHLGLRQGDCVALLMGNEPAYVWL
WLGLVKLGCAMACLNYNIRAKSLLHCFQCCGAKVLLVSPELQAAVEEILPSLKKDDVSIY
YVSRTSNTDGIDSFLDKVDEVSTEPIPESWRSEVTFSTPALYIYTSGTTGLPKAAMITHQ
RIWYGTGLTFVSGLKADDVIYITLPFYHSAALLIGIHGCIVAGATLALRTKFSASQFWDD
CRKYNVTVIQYIGELLRYLCNSPQKPNDRDHKVRLALGNGLRGDVWRQFVKRFGDICIYE
FYAATEGNIGFMNYARKVGAVGRVNYLQKKIITYDLIKYDVEKDEPVRDENGYCVRVPKG
EVGLLVCKITQLTPFNGYAGAKAQTEKKKLRDVFKKGDLYFNSGDLLMVDHENFIYFHDR
VGDTFRWKGENVATTEVADTVGLVDFVQEVNVYGVHVPDHEGRIGMASIKMKENHEFDGK
KLFQHIADYLPSYARPRFLRIQDTIEITGTFKHRKMTLVEEGFNPAVIKDALYFLDDTAK
MYVPMTEDIYNAISAKTLKL
|
|
|
|---|
| BDBM50168142 |
|---|
| n/a |
|---|
| Name | BDBM50168142 |
|---|
| Synonyms: | CHEMBL3716578 | US10849901, Compound 38 | US10953012, Example 9 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C25H17ClN4O3 |
|---|
| Mol. Mass. | 456.88 |
|---|
| SMILES | [O-][N+](=O)c1ccc(cc1)-c1cc(=O)n2nc(Cc3ccccc3)c(-c3ccc(Cl)cc3)c2[nH]1 |
|---|
| Structure | 
|
|---|
Search and Browse
