Reaction Details |
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Target | Cytosol aminopeptidase [33-68,L62W] |
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Ligand | BDBM50170884 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_1577950 (CHEMBL3806574) |
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Ki | 21100±n/a nM |
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Citation | Weglarz-Tomczak, E; Berlicki, L; Pawelczak, M; Nocek, B; Joachimiak, A; Mucha, A A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases. Eur J Med Chem117:187-96 (2016) [PubMed] Article |
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More Info.: | Get all data from this article, Assay Method |
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Cytosol aminopeptidase [33-68,L62W] |
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Name: | Cytosol aminopeptidase [33-68,L62W] |
Synonyms: | AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP) |
Type: | Enzyme |
Mol. Mass.: | 4015.44 |
Organism: | Sus scrofa (Pig) |
Description: | P28839[33-68,L62W] |
Residue: | 36 |
Sequence: | TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
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BDBM50170884 |
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n/a |
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Name | BDBM50170884 |
Synonyms: | CHEMBL3805495 |
Type | Small organic molecule |
Emp. Form. | C21H29N2O5P |
Mol. Mass. | 420.4391 |
SMILES | COc1ccc(CCNCC(N)P(O)(=O)CC(Cc2ccccc2)C(O)=O)cc1 |
Structure |
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