| Reaction Details |
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 | Report a problem with these data |
| Target | Free fatty acid receptor 3 |
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| Ligand | BDBM50200350 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1622016 (CHEMBL3864368) |
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| EC50 | >10000±n/a nM |
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| Citation |  Krasavin, M; Lukin, A; Bagnyukova, D; Zhurilo, N; Zahanich, I; Zozulya, S; Ihalainen, J; Forsberg, MM; Lehtonen, M; Rautio, J; Moore, D; Tikhonova, IG Free fatty acid receptor 1 (GPR40) agonists containing spirocyclic periphery inspired by LY2881835. Bioorg Med Chem24:5481-5494 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Free fatty acid receptor 3 |
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| Name: | Free fatty acid receptor 3 |
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| Synonyms: | FFAR3 | FFAR3_HUMAN | GPR41 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 38655.15 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1508992 |
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| Residue: | 346 |
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| Sequence: | MDTGPDQSYFSGNHWFVFSVYLLTFLVGLPLNLLALVVFVGKLQRRPVAVDVLLLNLTAS
DLLLLLFLPFRMVEAANGMHWPLPFILCPLSGFIFFTTIYLTALFLAAVSIERFLSVAHP
LWYKTRPRLGQAGLVSVACWLLASAHCSVVYVIEFSGDISHSQGTNGTCYLEFRKDQLAI
LLPVRLEMAVVLFVVPLIITSYCYSRLVWILGRGGSHRRQRRVAGLLAATLLNFLVCFGP
YNVSHVVGYICGESPAWRIYVTLLSTLNSCVDPFVYYFSSSGFQADFHELLRRLCGLWGQ
WQQESSMELKEQKGGEEQRADRPAERKTSEHSQGCGTGGQVACAES
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| BDBM50200350 |
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| n/a |
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| Name | BDBM50200350 |
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| Synonyms: | CHEMBL3926143 |
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| Type | Small organic molecule |
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| Emp. Form. | C34H42ClNO4 |
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| Mol. Mass. | 564.155 |
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| SMILES | Cl.Cc1ccc(CC2CCOC3(CCN(Cc4ccc(COc5ccc(CCC(O)=O)cc5)cc4)CC3)C2)cc1 |
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| Structure | 
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