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TargetMetalloproteinase inhibitor 3
LigandBDBM50225362
Substrate/Competitorn/a
Meas. Tech.ChEMBL_201218 (CHEMBL804012)
IC50>10000±n/a nM
Citation Nordmann, RWidmer, A Resolution and absolute configuration of the potent dopamine agonist N,N-diethyl-N'-[(3 alpha, 4a alpha, 10a beta)-1,2,3,4,4a,5,10,10a- -octahydro-6-hydroxy-1-propyl-3-benzo[g]quinolinyl]sulfamide. J Med Chem28:1540-2 (1985) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Metalloproteinase inhibitor 3
Name:Metalloproteinase inhibitor 3
Synonyms:TIMP3_RAT | Timp-3 | Timp3 | Tissue inhibitor of metalloproteinases 3 | Tissue inhibitor of metalloproteinases-3
Type:PROTEIN
Mol. Mass.:24241.51
Organism:Rattus norvegicus
Description:ChEMBL_10750
Residue:211
Sequence:
MTPWLGLVVLLSCWSLGHWGTEACTCSPSHPQDAFCNSDIVIRAKVVGKKLVKEGPFGTL
VYTIKQMKMYRGFSKMPHVQYIHTEASESLCGLKLEVNKYQYLLTGRVYEGKMYTGLCNF
VERWDHLTLSQRKGLNYRYHLGCNCKIKSCYYLPCFVTSKKECLWTDMLSNFGYPGYQSK
HYACIRQKGGYCSWYRGWAPPDKSISNATDP
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  Blast E-value cutoff:
BDBM50225362
n/a
NameBDBM50225362
Synonyms:Norprolac | QUINAGOLIDE
TypeSmall organic molecule
Emp. Form.C20H33N3O3S
Mol. Mass.395.559
SMILES[H][C@]12C[C@@H](CN(CCC)[C@]1([H])Cc1cccc(O)c1C2)NS(=O)(=O)N(CC)CC
Structure
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