| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor |
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| Ligand | BDBM50229871 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_138190 (CHEMBL747834) |
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| Kd | 1905±n/a nM |
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| Citation |  Bravo, P; Resnati, G; Angeli, P; Frigerio, M; Viani, F; Arnone, A; Marucci, G; Cantalamessa, F Synthesis and pharmacological evaluation of enantiomerically pure 4-deoxy-4-fluoromuscarines. J Med Chem35:3102-10 (1992) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Muscarinic acetylcholine receptor |
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| Name: | Muscarinic acetylcholine receptor |
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| Synonyms: | GPM3 | Muscarinic acetylcholine receptor M3 |
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| Type: | n/a |
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| Mol. Mass.: | 66272.13 |
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| Organism: | Cavia porcellus |
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| Description: | n/a |
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| Residue: | 587 |
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| Sequence: | MTLHSNSTTLPLFPNISTSWIHSPSEAGLPPGTVTHFGSYNISQAAGNFSSLNGTTSDPL
GGHTIWQVVFIAFLTGFLALVTIIGNILVIVSFKVNKQLKHVNNYFLLSLADLIIGVISM
NLFTTYIIMNRWALGNLACDLWLSIDYVASNASVMNLLVISFDRYFSITRPLTYRAKRTT
KRAGVMIGLAWVISFVLWAPAILFWQYFVGKRTVPPGECFIQFLSEPTITFGTAIAAFYM
PVTIMTILYWRIYKETEKRTKELAGLQASGTEAETENFVHPTGSSRSCSSYELQQQSLKH
SSRRKYSRCHFWFATKSWKPNAGQMDQDHSSSDSWNNYDAAASLENSASDEEDIGSETRA
IYSIVLKLPGHSTILNSTKLPSSDNLQVPEEDLEPMDMERNASKPQTQKSMDDGGSFQKS
FSNLPIQLESTMDTAKTSDANSSVSKTMATLPLSFKEATLAKRFALRTRSQITKRKRMSL
IKEKRAAQTLSAILLAFIITWTPYNIMVLVNTFCDSCIPKTYWNLGYWLCYINSTVNPVC
YALCNKTFRNTFKMLLLCQCDKRKRRKQQYQQRQSVIFHKRVPEQAL
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| BDBM50229871 |
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| n/a |
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| Name | BDBM50229871 |
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| Synonyms: | CHEMBL316804 |
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| Type | Small organic molecule |
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| Emp. Form. | C9H19FINO |
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| Mol. Mass. | 303.1561 |
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| SMILES | [I-].C[C@@H]1O[C@H](C[N+](C)(C)C)C[C@H]1F |
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| Structure | 
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