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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Mu-type opioid receptor | ||
| Ligand | BDBM83098 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEBML_1651389 | ||
| Ki | 18±n/a nM | ||
| Citation |  Prezzavento, O; Arena, E; Sánchez-Fernández, C; Turnaturi, R; Parenti, C; Marrazzo, A; Catalano, R; Amata, E; Pasquinucci, L; Cobos, EJ (+)-and (-)-Phenazocine enantiomers: Evaluation of their dual opioid agonist/s Eur J Med Chem125:603-610 (2017) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Mu-type opioid receptor | |||
| Name: | Mu-type opioid receptor | ||
| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO | ||
| Type: | Enzyme Catalytic Domain | ||
| Mol. Mass.: | 11165.58 | ||
| Organism: | GUINEA PIG | ||
| Description: | P97266 | ||
| Residue: | 98 | ||
| Sequence: |
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| BDBM83098 | |||
| n/a | |||
| Name | BDBM83098 | ||
| Synonyms: | (4R,4aS,7aR,12bS)-3-allyl-4a,9-dihydroxy-3-methyl-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-3-ium-7-one;iodide | (4R,4aS,7aR,12bS)-3-methyl-4a,9-bis(oxidanyl)-3-prop-2-enyl-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-3-ium-7-one;iodide | (4R,4aS,7aR,12bS)-4a,9-dihydroxy-3-methyl-3-prop-2-enyl-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-3-ium-7-one;iodide | MLS001334009 | Naloxone methiodide | SMR000875254 | cid_16219719 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C20H24NO4 | ||
| Mol. Mass. | 342.4083 | ||
| SMILES | C[N+]1(CC=C)CC[C@@]23[C@H]4Oc5c2c(C[C@@H]1[C@]3(O)CCC4=O)ccc5O | ||
| Structure | 
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