| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
|---|
| Ligand | BDBM84882 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 124±n/a nM |
|---|
| Comments | PDSP_928 |
|---|
| Citation |  Compton, DR; Rice, KC; De Costa, BR; Razdan, RK; Melvin, LS; Johnson, MR; Martin, BR Cannabinoid structure-activity relationships: correlation of receptor binding and in vivo activities. J Pharmacol Exp Ther265:218-26 (1993) [PubMed] |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Cannabinoid receptor 1 |
|---|
| Name: | Cannabinoid receptor 1 |
|---|
| Synonyms: | Brain-type cannabinoid receptor | CANNABINOID CB1 | CB-R | CB1 | CNR1_RAT | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cnr1 | Skr6 |
|---|
| Type: | G Protein-Coupled Receptor (GPCR) |
|---|
| Mol. Mass.: | 52856.55 |
|---|
| Organism: | Rattus norvegicus (rat) |
|---|
| Description: | P20272 |
|---|
| Residue: | 473 |
|---|
| Sequence: | MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNSPLVPAGDTTNITEFYNKSLSSFKENEENIQCGENFMDMECFMILNPSQQLAI
AVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFVDFHV
FHRKDSPNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCL
MWTIAIVIAVLPLLGWNCKKLQSVCSDIFPLIDETYLMFWIGVTSVLLLFIVYAYMYILW
KAHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPL
LAIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTA
QPLDNSMGDSDCLHKHANNTASMHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
|
|
|
|---|
| BDBM84882 |
|---|
| n/a |
|---|
| Name | BDBM84882 |
|---|
| Synonyms: | CAS_169742 | HHC, 9 beta-OH | HHC. 9 alpha-OH | NSC_169742 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H32O3 |
|---|
| Mol. Mass. | 332.477 |
|---|
| SMILES | CCCCCc1cc(O)c2C3CC(C)(O)CCC3C(C)(C)Oc2c1 |
|---|
| Structure | 
|
|---|
Search and Browse
