| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 4 |
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| Ligand | BDBM50007872 |
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| Substrate/Competitor | n/a |
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| Ki | 53.7±n/a nM |
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| Comments | PDSP_399 |
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| Citation |  Ansanay, H; Sebben, M; Bockaert, J; Dumuis, A Pharmacological comparison between [3H]GR 113808 binding sites and functional 5-HT4 receptors in neurons. Eur J Pharmacol298:165-74 (1996) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| 5-hydroxytryptamine receptor 4 |
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| Name: | 5-hydroxytryptamine receptor 4 |
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| Synonyms: | 5-HT-4 | 5-HT4 | 5-HT4L | 5-hydroxytryptamine receptor 4 | 5HT4R_MOUSE | Htr4 | Serotonin 4 (5-HT4) receptor | Serotonin receptor 4 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 43970.99 |
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| Organism: | MOUSE |
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| Description: | 5-HT4 HTR4 MOUSE::P97288 |
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| Residue: | 388 |
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| Sequence: | MDKLDANVSSNEGFRSVEKVVLLTFLAVVILMAILGNLLVMVAVCRDRQLRKIKTNYFIV
SLAFADLLVSVLVMPFGAIELVQDIWAYGEMFCLVRTSLDVLLTTASIFHLCCISLDRYY
AICCQPLVYRNKMTPLRIALMLGGCWVLPMFISFLPIMQGWNNIGIVDVIEKRKFSHNSN
STWCVFMVNKPYAITCSVVAFYIPFLLMVLAYYRIYVTAKEHAQQIQMLQRAGATSESRP
QPADQHSTHRMRTETKAAKTLCVIMGCFCFCWAPFFVTNIVDPFIDYTVPEQVWTAFLWL
GYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYKRPPILGQTVPCSTTTINGSTHVLRD
TVECGGQWESRCHLTATSPLVAAQPSDT
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| BDBM50007872 |
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| n/a |
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| Name | BDBM50007872 |
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| Synonyms: | 3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxylic acid (8-methyl-8-aza-bicyclo[3.2.1]oct-3-yl)-amide; hydrochloride | BIMU 1 | CHEMBL544755 | CHEMBL62023 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H24N4O2 |
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| Mol. Mass. | 328.4088 |
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| SMILES | CCn1c2ccccc2n(C(=O)NC2CC3CCC(C2)N3C)c1=O |TLB:12:13:20:16.17| |
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| Structure | 
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