| Reaction Details |
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 | Report a problem with these data |
| Target | Hrh3 protein |
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| Ligand | BDBM85023 |
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| Substrate/Competitor | n/a |
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| Ki | 0.15±n/a nM |
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| Comments | PDSP_885 |
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| Citation |  Brown, JD; O'Shaughnessy, CT; Kilpatrick, GJ; Scopes, DI; Beswick, P; Clitherow, JW; Barnes, JC Characterisation of the specific binding of the histamine H3 receptor antagonist radioligand [3H]GR168320. Eur J Pharmacol311:305-10 (1996) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Hrh3 protein |
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| Name: | Hrh3 protein |
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| Synonyms: | HISTAMINE H3 | HRH3 | Hrh3 protein |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 37860.96 |
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| Organism: | RAT |
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| Description: | Q5PPG3 |
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| Residue: | 344 |
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| Sequence: | MERAPPDGLMNASGTLAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFV
ADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCAS
SVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGG
SSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAG
PEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRGSKPSASSASLEKRMKMVSQSITQRF
RLSRDKKVAKSLAIIVSIFGLCWAPYTLLMIIRAACHGRCIPDY
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| BDBM85023 |
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| n/a |
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| Name | BDBM85023 |
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| Synonyms: | GR 168320 | GR-168320 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H25N5 |
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| Mol. Mass. | 275.3925 |
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| SMILES | NC(=NC1CCCCC1)N1CCC(CC1)c1cnc[nH]1 |w:2.2| |
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| Structure | 
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