| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 4 |
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| Ligand | BDBM85019 |
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| Substrate/Competitor | n/a |
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| Ki | 1.38±n/a nM |
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| Comments | PDSP_1604 |
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| Citation |  Claeysen, S; Sebben, M; Journot, L; Bockaert, J; Dumuis, A Cloning, expression and pharmacology of the mouse 5-HT(4L) receptor. FEBS Lett398:19-25 (1996) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| 5-hydroxytryptamine receptor 4 |
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| Name: | 5-hydroxytryptamine receptor 4 |
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| Synonyms: | 5-HT-4 | 5-HT4 | 5-HT4L | 5-hydroxytryptamine receptor 4 | 5HT4R_MOUSE | Htr4 | Serotonin 4 (5-HT4) receptor | Serotonin receptor 4 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 43970.99 |
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| Organism: | MOUSE |
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| Description: | 5-HT4 HTR4 MOUSE::P97288 |
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| Residue: | 388 |
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| Sequence: | MDKLDANVSSNEGFRSVEKVVLLTFLAVVILMAILGNLLVMVAVCRDRQLRKIKTNYFIV
SLAFADLLVSVLVMPFGAIELVQDIWAYGEMFCLVRTSLDVLLTTASIFHLCCISLDRYY
AICCQPLVYRNKMTPLRIALMLGGCWVLPMFISFLPIMQGWNNIGIVDVIEKRKFSHNSN
STWCVFMVNKPYAITCSVVAFYIPFLLMVLAYYRIYVTAKEHAQQIQMLQRAGATSESRP
QPADQHSTHRMRTETKAAKTLCVIMGCFCFCWAPFFVTNIVDPFIDYTVPEQVWTAFLWL
GYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYKRPPILGQTVPCSTTTINGSTHVLRD
TVECGGQWESRCHLTATSPLVAAQPSDT
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| BDBM85019 |
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| n/a |
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| Name | BDBM85019 |
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| Synonyms: | 4-Amino-5-chloro-N-(1-{4-[4-(dimethylamino)-1-piperidinyl]-4-oxobutyl}-3-methoxy-4-piperidinyl)-2-methoxybenzamide | RN 76186 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H40ClN5O4 |
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| Mol. Mass. | 510.069 |
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| SMILES | COC1CN(CCCC(=O)N2CCC(CC2)N(C)C)CCC1NC(=O)c1cc(Cl)c(N)cc1OC |
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| Structure | 
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