| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A1 |
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| Ligand | BDBM82557 |
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| Substrate/Competitor | n/a |
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| Ki | 4±n/a nM |
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| Comments | PDSP_945 |
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| Citation |  Hill, RJ; Oleynek, JJ; Hoth, CF; Kiron, MA; Weng, W; Wester, RT; Tracey, WR; Knight, DR; Buchholz, RA; Kennedy, SP Cloning, expression and pharmacological characterization of rabbit adenosine A1 and A3 receptors. J Pharmacol Exp Ther280:122-8 (1997) [PubMed] |
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| More Info.: | Get all data from this article |
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| Adenosine receptor A1 |
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| Name: | Adenosine receptor A1 |
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| Synonyms: | AA1R_RABIT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | ADORA1 | Adenosine receptor A1 (A1) |
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| Type: | Enzyme |
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| Mol. Mass.: | 36566.33 |
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| Organism: | Oryctolagus cuniculus (Rabbit) |
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| Description: | P34970 |
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| Residue: | 328 |
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| Sequence: | MPPSISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPETYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKAVVT
PRRAAVAIAGCWILSLVVGLTPMFGWNNLREVQRAWAANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRRQLSKKASASSGDPHKYYGKELKIAKSLALIL
FLFALSWLPLHILNCVTLFCPSCQKPSILVYTAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCRPAPAGDGDEDLPEEKPND
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| BDBM82557 |
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| n/a |
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| Name | BDBM82557 |
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| Synonyms: | I-ABA | IABA | N(6)-(4-Amino-3-iodobenzyl)adenosine |
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| Type | Small organic molecule |
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| Emp. Form. | C17H19IN6O4 |
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| Mol. Mass. | 498.275 |
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| SMILES | Nc1ccc(CNc2ncnc3n(cnc23)[C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)cc1I |
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| Structure | 
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