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TargetGamma-aminobutyric acid receptor subunit alpha-6
LigandBDBM85040
Substrate/Competitorn/a
Ki 1196±n/a nM
CommentsPDSP_1997
Citation Gunnersen, DKaufman, CMSkolnick, P Pharmacological properties of recombinant "diazepam-insensitive" GABAA receptors. Neuropharmacology35:1307-14 (1996) [PubMed]  Article
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Gamma-aminobutyric acid receptor subunit alpha-6
Name:Gamma-aminobutyric acid receptor subunit alpha-6
Synonyms:GABA A Alpha6Beta3Gamma2 | GABA A receptor alpha-6/beta-2/gamma-2 | GABA receptor alpha-6 subunit | GBRA6_RAT | Gabra-6 | Gabra6 | Gamma-aminobutyric acid receptor subunit alpha-6
Type:Enzyme Catalytic Domain
Mol. Mass.:51188.24
Organism:RAT
Description:GABA A Alpha6Beta2Gamma2 0 RAT::P30191
Residue:453
Sequence:
MLLLLPWLFSLLWIENAQAQLEDEGNFYSENVSRILDNLLEGYDNRLRPGFGGAVTEVKT
DIYVTSFGPVSDVEMEYTMDVFFRQTWTDERLKFKGPAEILSLNNLMVSKIWTPDTFFRN
GKKSIAHNMTTPNKLFRLMHNGTILYTMRLTINADCPMRLVNFPMDGHACPLKFGSYAYP
KSEIIYTWKKGPLYSVEVPEESSSLLQYDLIGQTVSSETIKSNTGEYVIMTVYFHLQRKM
GYFMIQIYTPCIMTVILSQVSFWINKESVPARTVFGITTVLTMTTLSISARHSLPKVSYA
TAMDWFIAVCFAFVFSALIEFAAVNYFTNLQSQKAERQAQTAAKPPVAKSKTTESLEAEI
VVHSDSKYHLKKRISSLTLPIVPSSEASKVLSRTPILPSTPVTPPLLLPAIGGTSKIDQY
SRILFPVAFAGFNLVYWIVYLSKDTMEVSSTVE
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BDBM85040
n/a
NameBDBM85040
Synonyms:CAS_123700 | NSC_123700 | ZK 91296
TypeSmall organic molecule
Emp. Form.C23H22N2O4
Mol. Mass.390.4318
SMILESCCOC(=O)c1ncc2[nH]c3cccc(OCc4ccccc4)c3c2c1COC
Structure
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