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TargetGalanin receptor type 2
LigandBDBM85073
Substrate/Competitorn/a
Ki 28±n/a nM
CommentsPDSP_3166
Citation Howard, ADTan, CShiao, LLPalyha, OCMcKee, KKWeinberg, DHFeighner, SDCascieri, MASmith, RGVan Der Ploeg, LHSullivan, KA Molecular cloning and characterization of a new receptor for galanin. FEBS Lett405:285-90 (1997) [PubMed]  Article
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Galanin receptor type 2
Name:Galanin receptor type 2
Synonyms:GALR2_RAT | Galanin R2 | Galanin receptor 2 | Galanin receptor type 2 | Galnr2 | Galr2
Type:Enzyme Catalytic Domain
Mol. Mass.:40697.04
Organism:RAT
Description:Galanin R2 GALR2 RAT::O08726
Residue:372
Sequence:
MNGSGSQGAENTSQEGGSGGWQPEAVLVPLFFALIFLVGTVGNALVLAVLLRGGQAVSTT
NLFILNLGVADLCFILCCVPFQATIYTLDDWVFGSLLCKAVHFLIFLTMHASSFTLAAVS
LDRYLAIRYPLHSRELRTPRNALAAIGLIWGLALLFSGPYLSYYRQSQLANLTVCHPAWS
APRRRAMDLCTFVFSYLLPVLVLSLTYARTLRYLWRTVDPVTAGSGSQRAKRKVTRMIII
VAVLFCLCWMPHHALILCVWFGRFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFR
KGFRKICAGLLRPAPRRASGRVSILAPGNHSGSMLEQESTDLTQVSEAAGPLVPPPALPN
CTASSRTLDPAC
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  Blast E-value cutoff:
BDBM85073
n/a
NameBDBM85073
Synonyms:CAS_3043476 | Galantide (M15) | NSC_3043476
TypeSmall organic molecule
Emp. Form.C23H30N2O3
Mol. Mass.382.4959
SMILESCOc1ccccc1N(CCOc1ccc(C)cc1)C(=O)CN1CCCCC1
Structure
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