| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Alpha-1A adrenergic receptor |
|---|
| Ligand | BDBM82564 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 144±n/a nM |
|---|
| Comments | PDSP_1655 |
|---|
| Citation |  Mos, J; Van Hest, A; Van Drimmelen, M; Herremans, AH; Olivier, B The putative 5-HT1A receptor antagonist DU125530 blocks the discriminative stimulus of the 5-HT1A receptor agonist flesinoxan in pigeons. Eur J Pharmacol325:145-53 (1997) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Alpha-1A adrenergic receptor |
|---|
| Name: | Alpha-1A adrenergic receptor |
|---|
| Synonyms: | adrenergic Alpha1 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 50699.64 |
|---|
| Organism: | pigeon |
|---|
| Description: | adrenergic Alpha1 0 pigeon::A0A1V4KJJ8 |
|---|
| Residue: | 464 |
|---|
| Sequence: | MAFLPGNSSDCSNCTHSVGPVNISKAILLGVILGGLIVFGVLGNILVILSVACHRHLQSV
THYYIINLAVADLLLTSTVLPFSATMEILGYWAFGRIFCNIWAAVDVLCCTASIMSLCII
SIDRYIGVSYPLRYPSIVTEKRGLLALLCVWALSLVISIGPLFGWKEPAPEDETICQITE
EPGYVLFSALGSFYLPLTIILVMYCRVYVVAKRENKGLSSGLKTERSHSEQVTLRIHRKN
APGASGSASNPKSKHHFSVRLLKFSREKKAAKTLGIVVGCFVLCWLPFFVVMPLGSFFPA
VKPPDTLFKITFWLGYLNSCINPIIYPCSSQEFKKAFQNVLRVQCLPRKQAAKKQSPSFN
LNHPASPSTESSRGVVRIPVGSGETFYKISKSDGVCEWKIFSAVQSMPAKTAVSKDCTAA
KVKSKGFLQECCCAGTSGNRGHENCKVPTIKIHTISLSESGEDV
|
|
|
|---|
| BDBM82564 |
|---|
| n/a |
|---|
| Name | BDBM82564 |
|---|
| Synonyms: | CAS_132787 | NSC_132787 | S 15535 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H24N2O2 |
|---|
| Mol. Mass. | 336.4275 |
|---|
| SMILES | C1C(Cc2ccccc12)N1CCN(CC1)c1cccc2OCCOc12 |
|---|
| Structure | 
|
|---|
Search and Browse
