Reaction Details |
| Report a problem with these data |
Target | Norepinephrine transporter |
---|
Ligand | BDBM22417 |
---|
Substrate/Competitor | n/a |
---|
Ki | 3.4±n/a nM |
---|
Comments | PDSP_1330 |
---|
Citation | Garreau, L; Emond, P; Belzung, C; Guilloteau, D; Frangin, Y; Besnard, JC; Chalon, S N-(3-lodoprop-2E-enyl)-2beta-carbomethoxy-3beta-(3',4'-dichloro phenyl)nortropane (beta-CDIT), a tropane derivative: pharmacological characterization as a specific ligand for the dopamine transporter in the rodent brain. J Pharmacol Exp Ther282:467-74 (1997) [PubMed] |
---|
More Info.: | Get all data from this article |
---|
|
Norepinephrine transporter |
---|
Name: | Norepinephrine transporter |
Synonyms: | n/a |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 2082.45 |
Organism: | RAT |
Description: | Norepinephrine transporter 0 RAT::Q9JIA2 |
Residue: | 19 |
Sequence: | |
BDBM22417 |
---|
n/a |
---|
Name | BDBM22417 |
Synonyms: | 3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine | CHEMBL295467 | LY 135252 | LY 94939 | LY135252 | LY139602 | Nisoxetine | Nisoxetine Inhibitor | US9944618, Compound ID No. 177 | [3-(2-methoxyphenoxy)-3-phenylpropyl](methyl)amine | [3H]Nisoxetine |
Type | radiolabeled ligand |
Emp. Form. | C17H21NO2 |
Mol. Mass. | 271.3541 |
SMILES | CNCCC(Oc1ccccc1OC)c1ccccc1 |
Structure |
|