| Reaction Details |
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 | Report a problem with these data |
| Target | Galanin receptor type 1 |
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| Ligand | BDBM50307254 |
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| Substrate/Competitor | n/a |
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| Ki | 4±n/a nM |
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| Comments | PDSP_1162 |
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| Citation |  Smith, KE; Forray, C; Walker, MW; Jones, KA; Tamm, JA; Bard, J; Branchek, TA; Linemeyer, DL; Gerald, C Expression cloning of a rat hypothalamic galanin receptor coupled to phosphoinositide turnover. J Biol Chem272:24612-6 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Galanin receptor type 1 |
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| Name: | Galanin receptor type 1 |
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| Synonyms: | GALR1_RAT | Galanin R1 | Galanin receptor type 1 | Galnr | Galnr1 | Galr1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 38883.91 |
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| Organism: | RAT |
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| Description: | Galanin R1 GALR1 RAT::Q62805 |
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| Residue: | 346 |
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| Sequence: | MELAPVNLSEGNGSDPEPPAEPRPLFGIGVENFITLVVFGLIFAMGVLGNSLVITVLARS
KPGKPRSTTNLFILNLSIADLAYLLFCIPFQATVYALPTWVLGAFICKFIHYFFTVSMLV
SIFTLAAMSVDRYVAIVHSRRSSSLRVSRNALLGVGFIWALSIAMASPVAYYQRLFHRDS
NQTFCWEHWPNQLHKKAYVVCTFVFGYLLPLLLICFCYAKVLNHLHKKLKNMSKKSEASK
KKTAQTVLVVVVVFGISWLPHHVIHLWAEFGAFPLTPASFFFRITAHCLAYSNSSVNPII
YAFLSENFRKAYKQVFKCRVCNESPHGDAKEKNRIDTPPSTNCTHV
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| BDBM50307254 |
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| n/a |
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| Name | BDBM50307254 |
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| Synonyms: | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40 |
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| Type | Small organic molecule |
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| Emp. Form. | C94H145N23O24 |
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| Mol. Mass. | 1981.2968 |
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| SMILES | CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O |r| |
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| Structure | 
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