| Reaction Details |
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 | Report a problem with these data |
| Target | Norepinephrine transporter |
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| Ligand | BDBM50069447 |
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| Substrate/Competitor | n/a |
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| Ki | 555±n/a nM |
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| Comments | PDSP_1303 |
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| Citation |  Owens, MJ; Morgan, WN; Plott, SJ; Nemeroff, CB Neurotransmitter receptor and transporter binding profile of antidepressants and their metabolites. J Pharmacol Exp Ther283:1305-22 (1997) [PubMed] |
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| More Info.: | Get all data from this article |
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| Norepinephrine transporter |
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| Name: | Norepinephrine transporter |
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| Synonyms: | n/a |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 2082.45 |
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| Organism: | RAT |
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| Description: | Norepinephrine transporter 0 RAT::Q9JIA2 |
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| Residue: | 19 |
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| Sequence: | |
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| BDBM50069447 |
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| n/a |
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| Name | BDBM50069447 |
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| Synonyms: | 1-(3-(4-(m-Chlorophenyl)-1-piperazinyl)propyl)-3-ethyl-4-(2-phenoxyethyl)-delta2-1,2,4-triazolin-5-one | 2-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-5-ethyl-4-(2-phenoxyethyl)-2,4-dihydro-3H-1,2,4-triazol-3-one | CHEMBL623 | NEFAZODONE | US9138393, Nefazodone HCl | US9144538, Nefazodone HCl |
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| Type | Small organic molecule |
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| Emp. Form. | C25H32ClN5O2 |
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| Mol. Mass. | 470.007 |
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| SMILES | CCc1nn(CCCN2CCN(CC2)c2cccc(Cl)c2)c(=O)n1CCOc1ccccc1 |
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| Structure | 
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