| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Galanin receptor type 2 |
|---|
| Ligand | BDBM85200 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 4.7±n/a nM |
|---|
| Comments | PDSP_857 |
|---|
| Citation |  Wang, S; He, C; Hashemi, T; Bayne, M Cloning and expressional characterization of a novel galanin receptor. Identification of different pharmacophores within galanin for the three galanin receptor subtypes. J Biol Chem272:31949-52 (1997) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Galanin receptor type 2 |
|---|
| Name: | Galanin receptor type 2 |
|---|
| Synonyms: | GALR2_RAT | Galanin R2 | Galanin receptor 2 | Galanin receptor type 2 | Galnr2 | Galr2 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 40697.04 |
|---|
| Organism: | RAT |
|---|
| Description: | Galanin R2 GALR2 RAT::O08726 |
|---|
| Residue: | 372 |
|---|
| Sequence: | MNGSGSQGAENTSQEGGSGGWQPEAVLVPLFFALIFLVGTVGNALVLAVLLRGGQAVSTT
NLFILNLGVADLCFILCCVPFQATIYTLDDWVFGSLLCKAVHFLIFLTMHASSFTLAAVS
LDRYLAIRYPLHSRELRTPRNALAAIGLIWGLALLFSGPYLSYYRQSQLANLTVCHPAWS
APRRRAMDLCTFVFSYLLPVLVLSLTYARTLRYLWRTVDPVTAGSGSQRAKRKVTRMIII
VAVLFCLCWMPHHALILCVWFGRFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFR
KGFRKICAGLLRPAPRRASGRVSILAPGNHSGSMLEQESTDLTQVSEAAGPLVPPPALPN
CTASSRTLDPAC
|
|
|
|---|
| BDBM85200 |
|---|
| n/a |
|---|
| Name | BDBM85200 |
|---|
| Synonyms: | Galanin (1-19), rat | Galanin rat |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C92H135N27O26 |
|---|
| Mol. Mass. | 2035.2216 |
|---|
| SMILES | CCC(C)C(NC(=O)C(C)NC(=O)C(Cc1cnc[nH]1)NC(=O)C1CCCN1C(=O)CNC(=O)C(CC(C)C)NC(=O)C(CC(C)C)NC(=O)C(Cc1ccc(O)cc1)NC(=O)CNC(=O)C(C)NC(=O)C(CO)NC(=O)C(CC(N)=O)NC(=O)C(CC(C)C)NC(=O)C(NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)CN)C(C)O)C(=O)NC(CC(O)=O)C(=O)NC(CC(N)=O)C(=O)NC(Cc1cnc[nH]1)C(N)=O |
|---|
| Structure | 
|
|---|
Search and Browse
