| Reaction Details |
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 | Report a problem with these data |
| Target | Galanin receptor type 3 |
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| Ligand | BDBM50307254 |
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| Substrate/Competitor | n/a |
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| Ki | 54±n/a nM |
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| Comments | PDSP_1162 |
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| Citation |  Wang, S; He, C; Hashemi, T; Bayne, M Cloning and expressional characterization of a novel galanin receptor. Identification of different pharmacophores within galanin for the three galanin receptor subtypes. J Biol Chem272:31949-52 (1997) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Galanin receptor type 3 |
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| Name: | Galanin receptor type 3 |
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| Synonyms: | GALR3_RAT | Galanin R3 | Galanin receptor type 3 | Galnr3 | Galr3 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40439.51 |
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| Organism: | RAT |
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| Description: | Galanin R3 GALR3 RAT::O88626 |
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| Residue: | 370 |
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| Sequence: | MADIQNISLDSPGSVGAVAVPVIFALIFLLGMVGNGLVLAVLLQPGPSAWQEPRSTTDLF
ILNLAVADLCFILCCVPFQAAIYTLDAWLFGAFVCKTVHLLIYLTMYASSFTLAAVSLDR
YLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDAR
RRALDVATFAAGYLLPVAVVSLAYGRTLCFLWAAVGPAGAAAAEARRRATGRAGRAMLAV
AALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYSLASRHFRA
RFRRLWPCGRRRHRHHHRAHRALRRVQPASSGPAGYPGDARPRGWSMEPRGDALRGGGET
RLTLSPRGPQ
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| BDBM50307254 |
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| n/a |
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| Name | BDBM50307254 |
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| Synonyms: | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40 |
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| Type | Small organic molecule |
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| Emp. Form. | C94H145N23O24 |
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| Mol. Mass. | 1981.2968 |
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| SMILES | CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O |r| |
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| Structure | 
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