| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Glutamate receptor |
|---|
| Ligand | BDBM50002369 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 1.41±n/a nM |
|---|
| Comments | PDSP_1011 |
|---|
| Citation |  Toms, NJ; Reid, ME; Phillips, W; Kemp, MC; Roberts, PJ A novel kainate receptor ligand [3H]-(2S,4R)-4-methylglutamate: pharmacological characterization in rabbit brain membranes. Neuropharmacology36:1483-8 (1997) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Glutamate receptor |
|---|
| Name: | Glutamate receptor |
|---|
| Synonyms: | Glutamate kainate | Glutamate-Kainate |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 96238.98 |
|---|
| Organism: | RABBIT |
|---|
| Description: | Glutamate-Kainate Glutamate kainate RABBIT::G1SXH9 |
|---|
| Residue: | 849 |
|---|
| Sequence: | MPNTTLTYDIQRINLFDSFEASRRACDQLALGVAALFGPSHSSSVSAVQSICNALEVPHI
QTRWKHPSVDNKDLFYINLYPDYAAISRAVLDLVLYYNWKTVTVVYEDSTGLIRLQELIK
APSRYNIKIKIRQLPSGNKDAKPLLKEMKKGKEFYVIFDCSHETAAEILKQILFMGMMTE
YYHYFFTTLDLFALDLELYRYSGVNMTGFRLLNIDNPHVSSIIEKWSMERLQAPPRPETG
LLDGMMTTEAALMYDAVYMVAIASHRASQLTVSSLQCHRHKPWRLGPRFMNLIKEAQWDG
LTGRITFNKTDGLRKNFDLDIISLKEEGTEKAAGEVSKHLYKVWKKIGIWNSNSGLNMTE
GNKDRSNNITDSLANRTLIVTTILEEPYVMYKKSDKPLYGNDRFEGYCLDLLKELSNILG
FIYDVKLVPDGKYGAQNDKGEWNGMVKELIDHKADLAVAPLTITYVREKVIDFSKPFMTL
GISILYRKPNGTNPGVFSFLNPLSPDIWMYVLLACLGVSCVLFVIARFTPYEWYNPHPCN
PDSDVVENNFTLLNSFWFGVGALMQQGSELMPKALSTRIVGGIWWFFTLIIISSYTANLA
AFLTVERMESPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQTA
LVKNNDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRD
KITIAILQLQEEGKLHMMKEKWWRGNGCPEEDNKEASALGVENIGGIFIVLAAGLVLSVF
VAIGEFIYKSRKNNDVEQCLSFNAIMEELGISLKNQKKLKKKSRTKGKSSFTSILTCHQR
RTQRKETVA
|
|
|
|---|
| BDBM50002369 |
|---|
| n/a |
|---|
| Name | BDBM50002369 |
|---|
| Synonyms: | (2S-(2alpha,3beta,4beta))-2-carboxy-4-(1-methylethenyl)-3-pyrrolidineacetic acid | (3S,4R)-3-(carboxymethyl)-4-(prop-1-en-2-yl)-L-proline | CHEMBL275040 | Digenin | Digensaeure | Helminal | Kainate | Kainsaeure | L-alpha-kainic acid | alpha-Kainic acid | digenic acid | kainic acid |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C10H15NO4 |
|---|
| Mol. Mass. | 213.2304 |
|---|
| SMILES | CC(=C)[C@H]1CN[C@@H]([C@H]1CC(O)=O)C(O)=O |r| |
|---|
| Structure | 
|
|---|
Search and Browse
