Reaction Details |
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Target | Melatonin receptor type 1A |
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Ligand | BDBM85065 |
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Substrate/Competitor | n/a |
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Ki | 933.25±n/a nM |
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Comments | PDSP_1123 |
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Citation | Beresford, IJ; Browning, C; Starkey, SJ; Brown, J; Foord, SM; Coughlan, J; North, PC; Dubocovich, ML; Hagan, RM GR196429: a nonindolic agonist at high-affinity melatonin receptors. J Pharmacol Exp Ther285:1239-45 (1998) [PubMed] |
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More Info.: | Get all data from this article |
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Melatonin receptor type 1A |
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Name: | Melatonin receptor type 1A |
Synonyms: | MTNR1A | MTR1A_PIG | Melatonin | Melatonin receptor type 1A |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 17908.30 |
Organism: | GUINEA PIG |
Description: | Melatonin 0 GUINEA PIG::O02781 |
Residue: | 154 |
Sequence: | YCYICHSLKYDRWYSNRNSLCCVFLICVLTLVAIVPNLCMGTLQYDPRIYSCTFAQSVSS
AYTIAVVVFHFLVPMVIVIFRYLRIWVLVLQIRWRAKPENNPRLKPQDFRNFVTMFVVFV
LFAICWAPLNFIGLAVASDPASMAPRIPEWLFVA
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BDBM85065 |
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n/a |
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Name | BDBM85065 |
Synonyms: | CAS_117946-91-5 | Luzindole | NSC_122162 |
Type | Small organic molecule |
Emp. Form. | C19H20N2O |
Mol. Mass. | 292.3749 |
SMILES | CC(=O)NCCc1c(Cc2ccccc2)[nH]c2ccccc12 |
Structure |
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