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TargetMelatonin receptor type 1A
LigandBDBM85065
Substrate/Competitorn/a
Ki 676.08±n/a nM
CommentsPDSP_1123
Citation Beresford, IJBrowning, CStarkey, SJBrown, JFoord, SMCoughlan, JNorth, PCDubocovich, MLHagan, RM GR196429: a nonindolic agonist at high-affinity melatonin receptors. J Pharmacol Exp Ther285:1239-45 (1998) [PubMed]
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Melatonin receptor type 1A
Name:Melatonin receptor type 1A
Synonyms:MTNR1A | MTR1A_PIG | Melatonin | Melatonin receptor type 1A
Type:Enzyme Catalytic Domain
Mol. Mass.:17908.30
Organism:GUINEA PIG
Description:Melatonin 0 GUINEA PIG::O02781
Residue:154
Sequence:
YCYICHSLKYDRWYSNRNSLCCVFLICVLTLVAIVPNLCMGTLQYDPRIYSCTFAQSVSS
AYTIAVVVFHFLVPMVIVIFRYLRIWVLVLQIRWRAKPENNPRLKPQDFRNFVTMFVVFV
LFAICWAPLNFIGLAVASDPASMAPRIPEWLFVA
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BDBM85065
n/a
NameBDBM85065
Synonyms:CAS_117946-91-5 | Luzindole | NSC_122162
TypeSmall organic molecule
Emp. Form.C19H20N2O
Mol. Mass.292.3749
SMILESCC(=O)NCCc1c(Cc2ccccc2)[nH]c2ccccc12
Structure
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