Reaction Details |
| Report a problem with these data |
Target | Melatonin receptor type 1A |
---|
Ligand | BDBM85065 |
---|
Substrate/Competitor | n/a |
---|
Ki | 251.18±n/a nM |
---|
Comments | PDSP_1123 |
---|
Citation | Beresford, IJ; Browning, C; Starkey, SJ; Brown, J; Foord, SM; Coughlan, J; North, PC; Dubocovich, ML; Hagan, RM GR196429: a nonindolic agonist at high-affinity melatonin receptors. J Pharmacol Exp Ther285:1239-45 (1998) [PubMed] |
---|
More Info.: | Get all data from this article |
---|
|
Melatonin receptor type 1A |
---|
Name: | Melatonin receptor type 1A |
Synonyms: | MTNR1A | MTNR1A protein | MTR1A_HUMAN | Mel-1A-R | Mel1a melatonin receptor | Melatonin 1A | Melatonin receptor | Melatonin receptor 1A | Melatonin receptor type 1 (MT1) | Melatonin receptor type 1A |
Type: | Enzyme |
Mol. Mass.: | 39392.94 |
Organism: | Homo sapiens (Human) |
Description: | P48039 |
Residue: | 350 |
Sequence: | MQGNGSALPNASQPVLRGDGARPSWLASALACVLIFTIVVDILGNLLVILSVYRNKKLRN
AGNIFVVSLAVADLVVAIYPYPLVLMSIFNNGWNLGYLHCQVSGFLMGLSVIGSIFNITG
IAINRYCYICHSLKYDKLYSSKNSLCYVLLIWLLTLAAVLPNLRAGTLQYDPRIYSCTFA
QSVSSAYTIAVVVFHFLVPMIIVIFCYLRIWILVLQVRQRVKPDRKPKLKPQDFRNFVTM
FVVFVLFAICWAPLNFIGLAVASDPASMVPRIPEWLFVASYYMAYFNSCLNAIIYGLLNQ
NFRKEYRRIIVSLCTARVFFVDSSNDVADRVKWKPSPLMTNNNVVKVDSV
|
|
|
BDBM85065 |
---|
n/a |
---|
Name | BDBM85065 |
Synonyms: | CAS_117946-91-5 | Luzindole | NSC_122162 |
Type | Small organic molecule |
Emp. Form. | C19H20N2O |
Mol. Mass. | 292.3749 |
SMILES | CC(=O)NCCc1c(Cc2ccccc2)[nH]c2ccccc12 |
Structure |
|