| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 2 |
|---|
| Ligand | BDBM82456 |
|---|
| Substrate/Competitor | n/a |
|---|
| Ki | 13.18±n/a nM |
|---|
| Comments | PDSP_376 |
|---|
| Citation |  Siehler, S; Seuwen, K; Hoyer, D [125I][Tyr3]octreotide labels human somatostatin sst2 and sst5 receptors. Eur J Pharmacol348:311-20 (1998) [PubMed] Article |
|---|
| More Info.: | Get all data from this article |
|---|
| |
| Somatostatin receptor type 2 |
|---|
| Name: | Somatostatin receptor type 2 |
|---|
| Synonyms: | SOMATOSTATIN SST2 | SRIF-1 | SS-2-R | SS2-R | SS2R | SSR2_HUMAN | SSTR2 | Somatostatin receptor type 2 (SSTR2) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 41344.94 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P30874 |
|---|
| Residue: | 369 |
|---|
| Sequence: | MDMADEPLNGSHTWLSIPFDLNGSVVSTNTSNQTEPYYDLTSNAVLTFIYFVVCIIGLCG
NTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMT
VDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMITMAVWGVSLLVILPIMIY
AGLRSNQWGRSSCTINWPGESGAWYTGFIIYTFILGFLVPLTIICLCYLFIIIKVKSSGI
RVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSMAISPTPALKGMFDFVVVL
TYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGTDDGERSDSKQDKSRLNETTETQRTL
LNGDLQTSI
|
|
|
|---|
| BDBM82456 |
|---|
| n/a |
|---|
| Name | BDBM82456 |
|---|
| Synonyms: | BIM 23030 | CAS_117580-24-2 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C45H57N9O8S2 |
|---|
| Mol. Mass. | 916.12 |
|---|
| SMILES | CC(C)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)CCSSC(NC1=O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r| |
|---|
| Structure | 
|
|---|
Search and Browse
