| Reaction Details |
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 | Report a problem with these data |
| Target | Galanin receptor type 3 |
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| Ligand | BDBM50273367 |
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| Substrate/Competitor | n/a |
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| Ki | 89.13±n/a nM |
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| Comments | PDSP_3165 |
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| Citation |  Smith, KE; Walker, MW; Artymyshyn, R; Bard, J; Borowsky, B; Tamm, JA; Yao, WJ; Vaysse, PJ; Branchek, TA; Gerald, C; Jones, KA Cloned human and rat galanin GALR3 receptors. Pharmacology and activation of G-protein inwardly rectifying K+ channels. J Biol Chem273:23321-6 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Galanin receptor type 3 |
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| Name: | Galanin receptor type 3 |
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| Synonyms: | GALR3_RAT | Galanin R3 | Galanin receptor type 3 | Galnr3 | Galr3 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40439.51 |
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| Organism: | RAT |
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| Description: | Galanin R3 GALR3 RAT::O88626 |
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| Residue: | 370 |
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| Sequence: | MADIQNISLDSPGSVGAVAVPVIFALIFLLGMVGNGLVLAVLLQPGPSAWQEPRSTTDLF
ILNLAVADLCFILCCVPFQAAIYTLDAWLFGAFVCKTVHLLIYLTMYASSFTLAAVSLDR
YLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDAR
RRALDVATFAAGYLLPVAVVSLAYGRTLCFLWAAVGPAGAAAAEARRRATGRAGRAMLAV
AALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYSLASRHFRA
RFRRLWPCGRRRHRHHHRAHRALRRVQPASSGPAGYPGDARPRGWSMEPRGDALRGGGET
RLTLSPRGPQ
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| BDBM50273367 |
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| n/a |
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| Name | BDBM50273367 |
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| Synonyms: | (2S,3S)-2-((S)-2-((S)-2-((S)-1-(2-((S)-2-((S)-2-((S)-2-(2-((S)-2-((S)-2-((S)-4-amino-2-((S)-2-((2S,3R)-2-((S)-2-(2-aminoacetamido)-3-(1H-indol-3-yl)propanamido)-3-hydroxybutanamido)-4-methylpentanamido)-4-oxobutanamido)-3-hydroxypropanamido)propanamido)acetamido)-3-(4-hydroxyphenyl)propanamido)-4-methylpentanamido)-4-methylpentanamido)acetyl)pyrrolidine-2-carboxamido)-3-(1H-imidazol-5-yl)propanamido)propanamido)-3-methylpentanoic acid | CHEMBL499980 | Galanin (1-16) | Galanin (1-16), porcine | Galanin (1-16), rat |
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| Type | Small organic molecule |
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| Emp. Form. | C78H116N20O21 |
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| Mol. Mass. | 1669.877 |
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| SMILES | CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(O)=O |r| |
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| Structure | 
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