| Reaction Details |
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 | Report a problem with these data |
| Target | Galanin receptor type 3 |
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| Ligand | BDBM85073 |
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| Substrate/Competitor | n/a |
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| Ki | 39.81±n/a nM |
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| Comments | PDSP_3166 |
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| Citation |  Smith, KE; Walker, MW; Artymyshyn, R; Bard, J; Borowsky, B; Tamm, JA; Yao, WJ; Vaysse, PJ; Branchek, TA; Gerald, C; Jones, KA Cloned human and rat galanin GALR3 receptors. Pharmacology and activation of G-protein inwardly rectifying K+ channels. J Biol Chem273:23321-6 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Galanin receptor type 3 |
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| Name: | Galanin receptor type 3 |
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| Synonyms: | GALNR3 | GALR3 | GALR3_HUMAN | Galanin R3 | Galanin receptor 3 | Galanin receptor type 3 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 39599.97 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Galanin R3 GALR3 HUMAN::O60755 |
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| Residue: | 368 |
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| Sequence: | MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLF
ILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDR
YLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDAR
RRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAV
AALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRA
RFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHG
GEAARGPE
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| BDBM85073 |
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| n/a |
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| Name | BDBM85073 |
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| Synonyms: | CAS_3043476 | Galantide (M15) | NSC_3043476 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H30N2O3 |
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| Mol. Mass. | 382.4959 |
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| SMILES | COc1ccccc1N(CCOc1ccc(C)cc1)C(=O)CN1CCCCC1 |
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| Structure | 
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