| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor M4 |
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| Ligand | BDBM82376 |
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| Substrate/Competitor | n/a |
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| Ki | 5.88±n/a nM |
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| Comments | PDSP_1795 |
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| Citation |  Chelala, JL; Kilani, A; Miller, MJ; Martin, RJ; Ernsberger, P Muscarinic receptor binding sites of the M4 subtype in porcine lung parenchyma. Pharmacol Toxicol83:200-7 (1998) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Muscarinic acetylcholine receptor M4 |
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| Name: | Muscarinic acetylcholine receptor M4 |
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| Synonyms: | CHRM4 | CHRM4 protein | Cholinergic, muscarinic M4 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 30028.84 |
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| Organism: | bovine |
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| Description: | A6QQE4 |
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| Residue: | 271 |
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| Sequence: | MTVLYVHISLASRSRVHKHRPEGPKEKKAKTLAFLKSPLMKQSVKKPPPPGDTTARGELR
NGKLEEAPPPVLPPPPRPMADKDTSNESSSGSATQNTKERPPTELSTTEATTPATPAPPL
QPRTLNPASKWSKIQIVTKQTGNECVTAIEIVPATPAGMRPAANVARKFASIARSQVRKK
RQMAARERKVTRTIFAILLAFILTWTPYNVMVLVNTFCQSCIPETVWSIGYWLCYVNSTI
NPACYALCNATFKKTFRHLLLCQYRNIGTAR
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| BDBM82376 |
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| n/a |
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| Name | BDBM82376 |
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| Synonyms: | CAS_80880-90-6 | NSC_5387 | TELENZEPINE |
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| Type | Small organic molecule |
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| Emp. Form. | C19H22N4O2S |
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| Mol. Mass. | 370.469 |
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| SMILES | CN1CCN(CC(=O)N2c3c(C)scc3C(=O)Nc3ccccc23)CC1 |
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| Structure | 
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