| Reaction Details |
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 | Report a problem with these data |
| Target | Gastrin-releasing peptide receptor |
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| Ligand | BDBM85498 |
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| Substrate/Competitor | n/a |
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| Ki | 6±n/a nM |
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| Comments | PDSP_1082 |
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| Citation |  Katsuno, T; Pradhan, TK; Ryan, RR; Mantey, SA; Hou, W; Donohue, PJ; Akeson, MA; Spindel, ER; Battey, JF; Coy, DH; Jensen, RT Pharmacology and cell biology of the bombesin receptor subtype 4 (BB4-R). Biochemistry38:7307-20 (1999) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| Gastrin-releasing peptide receptor |
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| Name: | Gastrin-releasing peptide receptor |
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| Synonyms: | GRPR_RAT | Gastrin-Releasing peptide | Gastrin-releasing peptide receptor | Grpr |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 43227.55 |
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| Organism: | RAT |
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| Description: | Gastrin-Releasing peptide 0 RAT::P52500 |
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| Residue: | 384 |
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| Sequence: | MDPNNCSHLNLEVDPFLSCNNTFNQTLSPPKMDNWFHPGIIYVIPAVYGLIIVIGLIGNI
TLIKIFCTVKSMRNVPNLFISSLALGDLLLLVTCAPVDASKYLADRWLFGRIGCKLIPFI
QLTSVGVSVFTLTALSADRYKAIVRPMDIQASHALMKICLKAALIWIVSMLLAIPEAVFS
DLHPFHVKDTNQTFISCAPYPHSNELHPKIHSMASFLVFYIIPLSIISVYYYFIARNLIQ
SAYNLPVEGNIHVKKQIESRKRLAKTVLVFVGLFAFCWLPNHVIYLYRSYHYSEVDTSML
HFITSICARLLAFTNSCVNPFALYLLSKSFRKQFNTQLLCCQPSLLNRSHSTGRSTTCMT
SFKSTNPSATFSLINGNICHEGYV
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| BDBM85498 |
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| n/a |
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| Name | BDBM85498 |
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| Synonyms: | CAS_5486808 | Litorin | NSC_5486808 |
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| Type | Small organic molecule |
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| Emp. Form. | C51H68N14O11S |
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| Mol. Mass. | 1085.238 |
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| SMILES | CSCCC(NC(=O)C(Cc1ccccc1)NC(=O)C(Cc1cnc[nH]1)NC(=O)CNC(=O)C(NC(=O)C(C)NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)C(CCC(N)=O)NC(=O)C1CCC(=O)N1)C(C)C)C(N)=O |
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| Structure | 
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